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CD 161

A potent, selective, orally bioavailable BET bromodomain inhibitor with IC50 of 7.2 and 28.2 nM for BRD4 BD2 and BRD4 BD1, respectively.

Product Specifications

CAS Number

1627716-22-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

435.487

Molecular Formula

C26H21N5O2

Notes

Research use only, not for human use.

Receptor

Bromodomain

Available Sizes

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