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PFI-2

A first-in-class, potent and selective inhibitor of SETD7 methyltransferase with Ki app/IC50 of 0.33/2 nM.

Product Specifications

CAS Number

1627676-59-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

499.5215

Molecular Formula

C23H25F4N3O3S

Notes

Research use only, not for human use.

Receptor

SETD7

Available Sizes

Frequently Asked Questions

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