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CPI-1205

A highly potent, selective EZH2 inhibitor with biochemical IC50 of 2 nM, cellular EC50 of 32 nM.

Product Specifications

CAS Number

1621862-70-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

518.57

Molecular Formula

C27H33F3N4O3

Notes

Research use only, not for human use.

Receptor

HMTase

Available Sizes

Curated Selection

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