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LY2857785

LY2857785 is a potenrt, reversible and ATP-competitive CDK9 inhibitor with IC50 of 11 nM, also inhibits CDK8 (IC50=16 nM) and weakly inhibits CSK7 (IC50=246 nM) .

Product Specifications

CAS Number

1619903-54-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

448.6036

Molecular Formula

C26H36N6O

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

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