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NU-2058

An ATP-competitive inhibitor of CDK1 and CDK2 with Ki of 5 uM and 12 uM respectively; inhibits human tumor cells with a mean GI50 of 13±7 uM.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

247.2963

Molecular Formula

C12H17N5O

Notes

Research use only, not for human use.

Receptor

CDK1|CDK2|TopoII

CAS Number

161058-83-9

Available Sizes

Curated Selection

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