THZ-1
A potent, selective, covalent CDK7 inhibitor with IC50 of 3.2 nM; also weakly inhibits CDK12 with IC50 of 250 nM; displays broad-based activity a subset of cancer cell lines with IC50s of <200 nM.
Product Specifications
CAS Number
1604810-83-4
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
566.0527
Molecular Formula
C31H28ClN7O2
Notes
Research use only, not for human use.
Receptor
CDK7
Available Sizes
Curated Selection
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