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PF-05387252

A potent, selective IRAK4 inhibitor with IC50 of 1.3 nM, 200-fold selectivity over IRAK1 (IC50=290 nM) .

Product Specifications

CAS Number

1604034-71-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

429.524

Molecular Formula

C25H27N5O2

Notes

Research use only, not for human use.

Receptor

IRAK

Available Sizes

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