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VX-984

VX-984 (M 9831) is a potent, selective inhibitor of DNA-PK with IC50 of 88±64 nM for inhibition of DNA-PKcs autophosphorylation (Ser2056) in A549 lung cancer cells.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

401.4702

Molecular Formula

C22H19D2N7O

Notes

Research use only, not for human use.

Receptor

DNA-PK

CAS Number

1562396-65-9

Available Sizes

Curated Selection

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