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SGC0946

SGC0946 is a highly potent and selective DOT1L methyltransferase inhibitor with IC50 of 0.3 nM; selectively kill mixed lineage leukaemia cells.

Product Specifications

CAS Number

1561178-17-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

618.57

Molecular Formula

C28H40BrN7O4

Notes

Research use only, not for human use.

Receptor

DOT1L

Available Sizes

Curated Selection

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