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TGR-1202 hydrochloride

TGR-1202 (RP5264, TGR1202, Umbralisib) is a potent, selective, orally available PI3Kδ inhibitor with IC50 of 22 nM.

Product Specifications

CAS Number

1532533-78-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

608.0101

Molecular Formula

C31H25ClF3N5O3

Notes

Research use only, not for human use.

Receptor

PI3K

Available Sizes

Frequently Asked Questions

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