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GSK 2981278

GSK 2981278 (GSK2981278) is a potent, highly selective RORγ/RORγt inhibitor that potently inhibits IL-17A and IL-22 protein secretion in human peripheral T cell with IC50 of 3.2 nM.

Product Specifications

CAS Number

1474110-21-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

461.617

Molecular Formula

C25H35NO5S

Notes

Research use only, not for human use.

Receptor

RORγ

Available Sizes

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