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Leucettamine B

Leucettamine B is a potent inhibitor of CLK1 (IC50=15 nM), Dyrk1A (IC50=40 nM), and Dyrk2 (IC50=35 nM) and a moderate inhibitor of CLK3 (IC50=4.5 uM) .

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

245.238

Molecular Formula

C12H11N3O3

Notes

Research use only, not for human use.

Receptor

CLK

CAS Number

147395-96-8

Available Sizes

Curated Selection

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