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Enasidenib

An orally available, selective, potent inhibitor of mutant IDH2 with IC50s of 100-400 nM for IDH2R140Q homodimer.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

473.375

Molecular Formula

C19H17F6N7O

Notes

Research use only, not for human use.

Receptor

IDH2

CAS Number

1446502-11-9

Available Sizes

Curated Selection

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