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PF-05089771

PF-05089771 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 11 nM.

Product Specifications

CAS Number

1430806-04-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

500.344

Molecular Formula

C18H12Cl2FN5O3S2

Notes

Research use only, not for human use.

Receptor

Na (V1.7) channel

Available Sizes

Curated Selection

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