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LY3039478

LY3039478 (Crenigacestat) is an exquisitely potent inhibitor of Notch-1 intracellular domain (N1ICD) cleavage with IC50 of 1 nM.

Product Specifications

CAS Number

1421438-81-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

464.4376

Molecular Formula

C22H23F3N4O4

Notes

Research use only, not for human use.

Receptor

Notch-1

Available Sizes

Curated Selection

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