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CAN-508

CAN-508 is a potent, selective CDK9 inhibitor with IC50 of 0.35 uM (CDK9/cyclin T1), displays >35 fold selectivity over CDK1/2/4/7 (IC50=13.5-70 uM) .

Product Specifications

CAS Number

140651-18-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

218.22

Molecular Formula

C9H10N6O

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

Curated Selection

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