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PFI-1

PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM in a cell-free assay.

Product Specifications

CAS Number

1403764-72-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

347.39

Molecular Formula

C16H17N3O4S

Notes

Research use only, not for human use.

Receptor

BRD2| BRD4

Available Sizes

Curated Selection

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