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S44819

S44819 (S-44819, Egis-1352 Afizagabar) is a novel potent, competitive, selective antagonist of the α5-GABAAR with Kd of 221 nM, IC50 of 585 nM (α5β2γ2) .

Product Specifications

CAS Number

1398496-82-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

365.382

Molecular Formula

C19H12FN3O2S

Notes

Research use only, not for human use.

Receptor

IGluR

Available Sizes

Frequently Asked Questions

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