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EPZ5676

EPZ-5676 is an S-adenosyl methionine (SAM) competitive inhibitor of protein methyltransferase DOT1L with Ki of 80 pM.

Product Specifications

CAS Number

1380288-87-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

562.71

Molecular Formula

C30H42N8O3

Notes

Research use only, not for human use.

Receptor

DOT1L

Available Sizes

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