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AGI-5198

AGI-5198 is the first highly potent and selective inhibitor of IDH1 R132H/R132C mutants with IC50 of 0.07 μM/0.16 μM.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

462.57

Molecular Formula

C27H31FN4O2

Notes

Research use only, not for human use.

Receptor

R132C-IDH1| R132H-IDH1

CAS Number

1355326-35-0

Available Sizes

Curated Selection

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