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SKI-2852

A highly potent, selective, and orally bioavailable 11β-HSD1 inhibitor with IC50 of 2.9 and 1.6 nM for hHSD1 and mHSD1, respectively.

Product Specifications

CAS Number

1346554-47-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

543.658

Molecular Formula

C27H34FN5O4S

Notes

Research use only, not for human use.

Receptor

11β-HSD

Available Sizes

Frequently Asked Questions

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