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PF-04136309

PF-4136309 (INCB8761) is a potent, selective, competitive, reversible full CCR2 antagonist with IC50 of 2-5 nM.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

568.59

Molecular Formula

C29H31F3N6O3

Notes

Research use only, not for human use.

Receptor

CCR2

CAS Number

1341224-83-6

Available Sizes

Curated Selection

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