PF-05190457
A potent, selective, and orally bioavailable ghrelin receptor (GHSR) inverse agonist with binding pKi of 8.36; displays excellent off-target activity in the CEREP panel at 10 uM with exception of serotonin 5-HT2B (IC50=3.7 uM) .
Product Specifications
CAS Number
1334782-79-4
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
512.676
Molecular Formula
C29H32N6OS
Notes
Research use only, not for human use.
Receptor
GHSR
Available Sizes
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