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GDC-0032

GDC-0032 is a potent, next-generation β isoform-sparing PI3K inhibitor targeting PI3Kα/δ/γ with IC50 of 0.29 nM/0.12 nM/0.97nM, >10 fold selective over PI3Kβ.

Product Specifications

CAS Number

1282512-48-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

460.53

Molecular Formula

C24H28N8O2

Notes

Research use only, not for human use.

Receptor

PI3Kα| PI3Kβ| PI3Kγ| PI3Kδ

Available Sizes

Curated Selection

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