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BIX02189

BIX02189 is a potent, selective inhibitor of MEK5 catalytic activity with IC50 of 1.5 nM, also inhibits ERK5 catalytic activity (IC50=59 nM) .

Product Specifications

CAS Number

1265916-41-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

440.5368

Molecular Formula

C27H28N4O2

Notes

Research use only, not for human use.

Receptor

MEK

Available Sizes

Curated Selection

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