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Delgocitinib

Delgocitinib (JTE-052, LEO 124249) is a potent, selective, orally active, pan-JAK inhibitor with IC50 of 2.8, 2.6, 13 and 58 nM for JAK1,2,3 and Tyk2, respectively.

Product Specifications

CAS Number

1263774-59-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

310.361

Molecular Formula

C16H18N6O

Notes

Research use only, not for human use.

Receptor

JAK

Available Sizes

Curated Selection

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