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UNC0638

A potent, selective, substrate-competitive inhibitor of G9a (EHMT2) and GLP (EHMT1) with IC50 of <15 nM and 19 nM in SAHH-coupled assays, respectively.

Product Specifications

CAS Number

1255580-76-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

509.7265

Molecular Formula

C30H47N5O2

Notes

Research use only, not for human use.

Receptor

G9a|GLP

Available Sizes

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