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(R) -DRF053 dihydrochloride

(R) -DRF053 dihydrochloride (DRF053) is a potent, cell-permeable, dual CK1/CDK inhibitor with IC50 of 14 nM, 220 nM and 80 nM for CK1, CDK5/p25 and CDK1/cyclin B, respectively.

Product Specifications

CAS Number

1241675-76-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

490.433

Molecular Formula

C23H29Cl2N7O

Notes

Research use only, not for human use.

Receptor

Casein Kinase

Available Sizes

Curated Selection

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