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APY0201

APY0201 is a potent, highly selective, ATP-competitive PIKfyve inhibitor (IC50=5.2 nM) that interrupts the conversion of phosphatidylinositol 3-phosphate (PtdIns3P) to PtdIns (3,5) P2.

Product Specifications

CAS Number

1232221-74-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

413.48

Molecular Formula

C23H23N7O

Notes

Research use only, not for human use.

Receptor

PIKfyve

Available Sizes

Frequently Asked Questions

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