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URMC-099

URMC-099 is a potent, orally bioavailable, brain penetrant inhibitor of mixed lineage kinase 3 (MLK3) with IC50 of 14 nM.

Product Specifications

CAS Number

1229582-33-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

421.5368

Molecular Formula

C27H27N5

Notes

Research use only, not for human use.

Receptor

Abl1|AuroraA|AuroraB|AuroraC|CDK1|CDK2|c-Met|DLK|IGF-1R|InsulinReceptor|Lck|LRRK2|MEKK2|MLK1|MLK2|MLK3|ROCK1|ROCK2|SGK|SGK1|Syk|TrkA|TrkB|VEGFR1/FLT1

Available Sizes

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