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XE-991

XE-991 is a potent, selective and orally active blocker of voltage-gated potassium channels Kv7 (KCNQ) that blocks KCNQ1, KCNQ2 and KCNQ2+KCNQ3 with Kd of 0.78, 0.7 and 0.6 uM, respectively.

Product Specifications

CAS Number

122955-42-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

376.45

Molecular Formula

C26H20N2O

Notes

Research use only, not for human use.

Receptor

Potassium Channel

Available Sizes

Curated Selection

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