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Sapanisertib

Sapanisertib (INK-128, MLN0128) is a potent, ATP-competitive, orally active dual mTORC1/2 inhibitor with Ki of 1.4 nM in cell-free assays.

Product Specifications

CAS Number

1224844-38-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

309.33

Molecular Formula

C15H15N7O

Notes

Research use only, not for human use.

Receptor

MTOR|PI3Kα|PI3Kγ|PI3Kδ

Available Sizes

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