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LOXO-101 sulfate

LOXO-101 (ARRY-470, Larotrectinib) is potent, selective pan-TRK inhibitor with cellular IC50 of 2-20 nM against TRKA, TRKB, and TRKC kinases.

Product Specifications

CAS Number

1223405-08-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

526.5137

Molecular Formula

C21H24F2N6O6S

Notes

Research use only, not for human use.

Receptor

Trk

Available Sizes

Frequently Asked Questions

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