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Apatinib Mesylate

Apatinib (YN968D1) is a multitargeted tyrosine kinase inhibitor (TKI) that inhibits VEGFR-2 (Flk-1/KDR, IC50=1 nM), RET, c-Kit and c-Src (IC50=13, 429 and 530 nM respectively) .

Product Specifications

CAS Number

1218779-75-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

493.58

Molecular Formula

C25H27N5O4S

Notes

Research use only, not for human use.

Receptor

VEGFR2|RET

Available Sizes

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