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SB 206553

SB 206553 is a potent and selective 5-HT2B/5-HT2C receptor antagonist with pA2 of 8.89 for rat 5-HT2B, pKi of 7.92 for human 5-HT2C, displays >80-fold selectivity over other 5-HT receptor subtypes.

Product Specifications

CAS Number

1197334-04-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

328.8

Molecular Formula

C17H16N4O.HCl

Notes

Research use only, not for human use.

Receptor

5-HT Receptor

Available Sizes

Curated Selection

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