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TAK-259 hydrochloride

A potent and selective human α1D adrenoceptor (α1D-AR) antagonist with Ki of 1.1 nM; displays 200-fold and 800-fold selectivity against α1A- and α1B-AR, respectively.

Product Specifications

CAS Number

1192347-42-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

410.694

Molecular Formula

C14H14Cl3N3O3S

Notes

Research use only, not for human use.

Receptor

Adrenergic Receptor

Available Sizes

Curated Selection

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