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MK-8617

A potent, orally active pan-inhibitor of HIF prolyl hydroxylase (HIF-PHD) with IC50 of 1.0,1.0, and 14 nM for HIF-PHD1, 2, and 3, respectively.

Product Specifications

CAS Number

1187990-87-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

443.45

Molecular Formula

C24H21N5O4

Notes

Research use only, not for human use.

Receptor

PHD1|PHD2|PHD3|PHD1, PHD2, PHD3

Available Sizes

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