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MK2 inhibitor III

A potent, cell-permeable inhibitor of MK2 with IC50 of 8.5 nM; less potently blocks MK3 and MK5 (IC50s=210 and 81 nM, respectively) .

Product Specifications

CAS Number

1186648-22-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

358.4

Molecular Formula

C21H16N4O • H2O

Notes

Research use only, not for human use.

Receptor

MAPKAPK2 (MK2)

Available Sizes

Curated Selection

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