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PF-8380

Potent autotaxin inhibitor (IC50 = 2.8 nM in isolated enzyme assay; 101 nM in human whole blood) .

Product Specifications

CAS Number

1144035-53-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

478.33

Molecular Formula

C22H21Cl2N3O5

Notes

Research use only, not for human use.

Receptor

Autotaxin

Available Sizes

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