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Edicotinib

Edicotinib (JNJ 40346527, PRV 6527) is a potent, selective, orally bioavailable CSF-1R inhibitor with IC50 of 3.2 nM; shows weak affinity for KIT and FLT3 (IC50= 20 nM and 190 nM, respectively) .

Product Specifications

CAS Number

1142363-52-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

461.61

Molecular Formula

C27H35N5O2

Notes

Research use only, not for human use.

Receptor

CSF1R

Available Sizes

Curated Selection

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