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E7449

E7449 (2X-121) is a potent, orally bioavailable, brain penetrable dual inhibitor of PARP1/2 and TNKS1/2 with IC50 of 2.0/1.0 nM (PARP1/2), 50-100 nM (TNKS1/2) .

Product Specifications

CAS Number

1140964-99-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

317.3446

Molecular Formula

C18H15N5O

Notes

Research use only, not for human use.

Receptor

PARP

Available Sizes

Curated Selection

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