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Cabozantinib (S-malate)

Cabozantinib (XL184) is a potent, multi-kinase inhibitor that inhibits VEGFR2, c-Met, Kit, Axl and Flt3 with IC50 of 0.035, 1.3, 4.6, 7 and 11.3 nM, respectively.

Product Specifications

CAS Number

1140909-48-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

635.5931

Molecular Formula

C32H30FN3O10

Notes

Research use only, not for human use.

Receptor

AXL|c-Met|Kit|VEGFR2/KDR|VEGFR3/FLT4

Available Sizes

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