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Mirogabalin besylate

Mirogabalin besylate (DS-5565) is a novel potent, selective ligand of the α2δ subunit of voltage-gated calcium channels with Kd of 13.5/22.7/27.0/47.6 nM for huamn α2δ-1, human α2δ-2, rat α2δ-1 and rat α2δ-2 subunits, respectively.

Product Specifications

CAS Number

1138245-21-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

367.46

Molecular Formula

C18H25NO5S

Notes

Research use only, not for human use.

Receptor

Calcium Channel

Available Sizes

Frequently Asked Questions

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