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Entrectinib

Entrectinib (NMS-E628, RXDX-101, NMS-01191372) is a potent, ATP-competitive, orally available pan-TRK, ROS1 and ALK inhibitor with IC50 of 1/3/5/12/7 nM for TRKA/TRKB/TRKC/ALK/ROS1, respectively.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

560.6375

Molecular Formula

C31H34F2N6O2

Notes

Research use only, not for human use.

Receptor

ALK|ROS1|TrkA|TrkB|TrkC

CAS Number

1108743-60-7

Available Sizes

Curated Selection

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