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CI-966

CI-966 (PD 126141) is a potent, selective inhibitor of the GABA transporter GAT-1 with IC50 of 0.26 and 1.2 uM for human and rat GAT-1, respectively.

Product Specifications

CAS Number

110283-79-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

473.415

Molecular Formula

C23H21F6NO3

Notes

Research use only, not for human use.

Receptor

GAT

Available Sizes

Curated Selection

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