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BIX02188 (c)

BIX02188 is a selective inhibitor of MEK5 with IC50 of 4.3 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

412.48

Molecular Formula

C25H24N4O2

Notes

Research use only, not for human use.

Receptor

ERK5| MEK1| MEK2| MEK5| TGFβR1

CAS Number

1094614-84-2

Available Sizes

Curated Selection

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