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IT1t dihydrochloride

A highly potent, selective, orally bioavailable CXCR4 inhibitor with binding IC50 of 8 nM for hCXCR4, IC50 of 1.1 nM in Ca2+-mobilization assays.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

479.57334

Molecular Formula

C21H36Cl2N4S2

Notes

Research use only, not for human use.

Receptor

Chemokine Receptor

CAS Number

1092776-63-0

Available Sizes

Curated Selection

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