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GSK-923295

The first potent, allosteric inhibitor of CENP-E kinesin motor ATPase activity with Ki of 3.2 nM.

Product Specifications

CAS Number

1088965-37-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

592.1282

Molecular Formula

C32H38ClN5O4

Notes

Research use only, not for human use.

Receptor

CENP-E

Available Sizes

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