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Lifitegrast

A potent LFA-1/ICAM-1 antagonist with IC50 of 9 nM in HuT78 cells; exhibits good in vitro safety profile and low potency on CYP3A4, CYP2C9 and hERG.

Product Specifications

CAS Number

1025967-78-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

615.4811

Molecular Formula

C29H24Cl2N2O7S

Notes

Research use only, not for human use.

Receptor

LFA-1

Available Sizes

Curated Selection

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