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Fostamatinib

Fostamatinib (R788 disodium salt) is a prodrug of the active metabolite R406, which is a potent, ATP-competitive inhibitor of Syk kinase with Ki/IC50 of 30/41 nM.

Product Specifications

CAS Number

1025687-58-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

624.4232

Molecular Formula

C23H24FN6Na2O9P

Notes

Research use only, not for human use.

Receptor

Syk

Available Sizes

Frequently Asked Questions

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